SCHEMBL14224712

SCHEMBL14224712

C=C1C(=O)N(c2ccc(SC(F)(F)F)cc2)C(=O)N1Cc1ccnc(NC(=O)CN(C)CCN(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 19/20 0.51
HCK P08631 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076749 0.85 IGF1R (0.67) IGF1RMAPK14
SCHEMBL2936805 0.83 IGF1R (0.74) IGF1R
SCHEMBL14214983 0.80 IGF1R (0.54) IGF1R
SCHEMBL14224713 0.79 IGF1R (0.50) IGF1R
SCHEMBL14224724 0.77 IGF1R (0.46) IGF1R
SCHEMBL13077177 0.77 IGF1R (0.46) IGF1R
SCHEMBL2934755 0.77 IGF1R (0.73) IGF1R
SCHEMBL31572879 0.76 IGF1R (0.80) IGF1R
SCHEMBL13076750 0.76 IGF1R (0.62) IGF1R
SCHEMBL13076351 0.75 IGF1R (0.51) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7354933-B2 Protein kinase inhibitors; antitumor agents; such as 5-methyl-1-quinol-4-ylmethyl-3-(4-trifluoromethanesulfonylphenyl)imidazolidine-2,4-dione trifluoroacetate AVENTIS PHARMA SA (FR) 2008-04-08 US disclosed