SCHEMBL1423896

SCHEMBL1423896

COc1ccc(-c2cnn3ccc(NC4CCC(N)CC4)nc23)cc1OC

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 15/20 0.70
PIM2 Q9P1W9 12/20 0.70
PIK3CG P48736 1/20 0.58
FYN P06241 1/20 0.55
MAPT P10636 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
KMT2A Q03164 1/20 0.52
FLT3 P36888 3/20 0.52
RET P07949 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423893 1.00 PIM1 (0.70) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1424084 0.90 PIK3CG (0.71) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1424085 0.90 PIK3CG (0.71) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1423993 0.87 PIM1 (0.68) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1423991 0.87 PIM1 (0.68) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1424538 0.87 PIK3CG (0.57) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1424537 0.87 PIK3CG (0.57) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1424076 0.84 PIM1 (0.71) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL1423761 0.84 PIM1 (0.71) PIM1PIM2PIK3CGFYNMAPT
SCHEMBL4328408 0.82 PIK3CG (0.72) PIM1PIM2PIK3CGMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081933-B1 PYRAZOLOPYRIMIDINES AS PI3K LIPID KINASE INHIBITORS NOVARTIS AG (CH) 2011-03-23 EP claimed
US-20090286779-A1 PYRAZOLOPYRIMIDINES AS LIPID KINASE INHIBITORS NOVARTIS AG 2009-11-19 US claimed
EP-2081933-B1 PYRAZOLOPYRIMIDINES AS PI3K LIPID KINASE INHIBITORS NOVARTIS AG (CH) 2011-03-23 EP disclosed
US-20090286779-A1 PYRAZOLOPYRIMIDINES AS LIPID KINASE INHIBITORS NOVARTIS AG 2009-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286779-A1 PYRAZOLOPYRIMIDINES AS LIPID KINASE INHIBITORS ATR, ATM, CHEK1 PIM1 452/4885PIM2 846/4885PIK3CG 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.