SCHEMBL1423946

SCHEMBL1423946

O=C(c1ccc(-n2nc(C(F)(F)F)c3c2CCOC3)cc1)N1CC(O)C1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 15/20 0.67
CYP2D6 P10635 5/20 0.58
CYP2C9 P11712 7/20 0.50
CYP1A2 P05177 4/20 0.50
GAA P10253 1/20 0.49
CYP2C19 P33261 3/20 0.45
UGCG Q16739 1/20 0.43
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423620 0.92 GRIA2 (0.65) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423747 0.88 GRIA2 (0.81) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423653 0.88 GRIA2 (0.84) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423711 0.87 GRIA2 (0.66) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL3143259 0.86 GRIA2 (0.78) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1424200 0.85 GRIA2 (0.54) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423813 0.85 GRIA2 (0.62) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL13300519 0.84 GRIA2 (0.71) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423867 0.80 GRIA2 (1.00) GRIA2CYP2D6CYP2C9CYP1A2GAA
SCHEMBL1423623 0.80 GRIA2 (0.96) GRIA2CYP2D6CYP2C9CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086643-B1 COMPOUNDS WHICH POTENTIATE AMPA RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LTD (GB) 2011-03-23 EP disclosed
US-20100137276-A1 COMPOUNDS WHICH POTENTIATE AMPA RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED 2010-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137276-A1 COMPOUNDS WHICH POTENTIATE AMPA RECEPTOR AND USES THEREOF IN MEDICINE GRIN1, GRM2, GRIN3A GRIA2 23/4885CYP2D6 1687/4885CYP2C9 2591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.