SCHEMBL14291981

SCHEMBL14291981

Cc1nn(-c2ccc(C#N)c(NC3CCOCC3)c2)c(N)c1N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.43
HSP90AB1 P08238 2/20 0.43
IRAK4 Q9NWZ3 2/20 0.36
TTK P33981 2/20 0.36
PRKCQ Q04759 1/20 0.35
PRKCD Q05655 1/20 0.35
MBOAT4 Q96T53 1/20 0.35
TBK1 Q9UHD2 4/20 0.35
JAK2 O60674 1/20 0.35
AR P10275 3/20 0.34
LRRK2 Q5S007 1/20 0.34
BRD4 O60885 1/20 0.34
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4581038 0.92 HSP90AA1 (0.43) HSP90AA1HSP90AB1IRAK4TTKPRKCQ
SCHEMBL4580224 0.78 HSP90AA1 (0.42) HSP90AA1HSP90AB1IRAK4TTKPRKCQ
SCHEMBL4581830 0.78 HSP90AA1 (0.41) HSP90AA1HSP90AB1IRAK4TTKPRKCQ
SCHEMBL4581868 0.71 HSP90AA1 (0.64) HSP90AA1HSP90AB1
SCHEMBL3628058 0.71 HSP90AB1 (0.65) HSP90AA1HSP90AB1
SCHEMBL3628057 0.71 HSP90AB1 (0.65) HSP90AA1HSP90AB1
SCHEMBL421243 0.71 HSP90AA1 (0.62) HSP90AA1
SCHEMBL14177807 0.70 MAPT (0.46) ARKMT2A
SCHEMBL4581082 0.70 PRKCQ (0.40) IRAK4PRKCQPRKCDTBK1JAK2
SCHEMBL4580776 0.69 PRKCQ (0.43) IRAK4PRKCQPRKCDJAK2LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008024978-A2 TETRAHYDROINDOLONE AND TETRAHYDROINDAZOLONE DERIVATIVES SERENEX, INC. (US) 2008-02-28 WO disclosed