SCHEMBL14306579

SCHEMBL14306579

CCn1c(=O)c(-c2cccs2)cc2c(C)nc(Nc3ccc(N4CCNCC4)cc3)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 16/20 0.46
CCND1 P24385 16/20 0.46
CCND2 P30279 13/20 0.46
CCND3 P30281 13/20 0.46
WEE1 P30291 1/20 0.45
CCNA2 P20248 8/20 0.45
CDK2 P24941 8/20 0.45
CCNA1 P78396 5/20 0.45
CCNE2 O96020 4/20 0.45
CCNE1 P24864 4/20 0.45
CCNB2 O95067 3/20 0.45
CDK1 P06493 3/20 0.45
CCNB1 P14635 3/20 0.45
CCNB3 Q8WWL7 3/20 0.45
FGFR1 P11362 5/20 0.44
FGFR2 P21802 5/20 0.44
FGFR4 P22455 5/20 0.44
FGFR3 P22607 5/20 0.44
PAK1 Q13153 3/20 0.43
PAK3 O75914 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL189156 0.92 WEE1 (0.54) CDK4CCND1CCND2CCND3WEE1
SCHEMBL188946 0.91 WEE1 (0.47) CDK4CCND1CCND2CCND3WEE1
SCHEMBL4225936 0.87 CDK4 (0.47) CDK4CCND1CCND2CCND3WEE1
SCHEMBL189185 0.87 WEE1 (0.46) CDK4CCND1CCND2CCND3WEE1
SCHEMBL4352016 0.85 WEE1 (0.44) CDK4CCND1CCND2CCND3WEE1
SCHEMBL189897 0.83 KDM4E (0.57) CDK4CCND1CCND2CCND3CCNA2
SCHEMBL14300938 0.83 PIK3CD (0.58) CDK4CCND1CCND2CCND3WEE1
SCHEMBL189076 0.81 CDK4 (0.42) CDK4CCND1CCND2CCND3WEE1
SCHEMBL3338688 0.79 CDK4 (0.56) CDK4CCND1CCND2CCND3CCNA2
SCHEMBL189768 0.78 HSD17B10 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021389-A2 USING PI3K AND MEK MODULATORS IN TREATMENTS OF CANCER EXELIXIS, INC. (US) 2008-02-21 WO disclosed