SCHEMBL14307347

SCHEMBL14307347

Bc1ccc(Cn2cc(C(=O)O)c(=O)c3c(F)ccc(F)c32)c(F)c1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 12/20 0.58
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
STAT3 P40763 1/20 0.37
MAPT P10636 1/20 0.35
TP53 P04637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2486523 0.86 CHRM1 (0.58) CHRM1ALDH1A1HTT
SCHEMBL2486081 0.84 CHRM1 (0.76) CHRM1ALDH1A1HTTMAPT
SCHEMBL2486292 0.81 CHRM1 (0.58) CHRM1ALDH1A1HTT
SCHEMBL2881808 0.81 CHRM1 (0.70) CHRM1ALDH1A1HTTMAPTLMNA
SCHEMBL2486353 0.80 CHRM1 (0.57) CHRM1ALDH1A1HTTTP53RXFP1
SCHEMBL2487845 0.80 CHRM1 (0.57) CHRM1ALDH1A1HTT
SCHEMBL2487841 0.78 CHRM1 (0.55) CHRM1ALDH1A1HTT
SCHEMBL2487906 0.78 CHRM1 (0.60) CHRM1ALDH1A1
SCHEMBL14308113 0.78 CHRM1 (0.56) CHRM1ALDH1A1HTTMAPTLMNA
SCHEMBL2488977 0.78 CHRM1 (0.55) CHRM1ALDH1A1MAPTTP53RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008002621-A2 BENZYL-SUBSTITUTED QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2008-01-03 WO disclosed