SCHEMBL14319080

SCHEMBL14319080

Cc1ccc(Nc2ncc(C(=O)NC3CCCC3)c(C(F)(F)F)n2)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 15/20 0.55
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
CYP2C9 P11712 5/20 0.49
CYP1A2 P05177 5/20 0.49
CYP3A4 P08684 4/20 0.49
LRRK2 Q5S007 4/20 0.49
CYP2C19 P33261 3/20 0.49
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3382316 0.90 CNR2 (0.66) CNR2RAB9ACYP2C9CYP1A2CYP3A4
SCHEMBL3380444 0.90 CNR2 (0.65) CNR2RAB9ACYP2C9CYP1A2CYP3A4
SCHEMBL3383233 0.89 CNR2 (0.66) CNR2RAB9ACYP2C9CYP1A2CYP3A4
SCHEMBL3379871 0.85 CNR2 (0.70) CNR2CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL13070075 0.84 CNR2 (0.71) CNR2CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL3380632 0.83 CNR2 (0.53) CNR2CYP2C9CYP1A2CYP3A4LRRK2
SCHEMBL3380625 0.83 CNR2 (0.66) CNR2CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL3377534 0.83 CNR2 (0.66) CNR2CYP2C9CYP1A2CYP3A4LRRK2
SCHEMBL13503356 0.82 CNR2 (0.76) CNR2CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL13503363 0.82 CNR2 (0.63) CNR2CYP2C9CYP1A2CYP3A4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878725-A2 Pyrimidine derivatives and their use as CB2 modulators GLAXO GROUP LIMITED (GB) 2008-01-16 EP disclosed