SCHEMBL14345728

SCHEMBL14345728

CCc1nc(=O)c(C)c2n1CCc1c-2[nH]c2ccc(OC)cc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.62
CYP1A1 P04798 8/20 0.62
CYP1B1 Q16678 8/20 0.62
KDM4E B2RXH2 6/20 0.62
MAPT P10636 4/20 0.62
ALDH1A1 P00352 3/20 0.62
NPC1 O15118 2/20 0.62
POLB P06746 2/20 0.62
RAB9A P51151 2/20 0.62
KMT2A Q03164 2/20 0.62
HPGD P15428 2/20 0.62
ESR1 P03372 1/20 0.62
TP53 P04637 1/20 0.62
NFKB1 P19838 1/20 0.62
NFKB2 Q00653 1/20 0.62
RELA Q04206 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
PDE5A O76074 3/20 0.52
ALOX15 P16050 2/20 0.51
TDP1 Q9NUW8 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14345707 0.89 CYP1A2 (0.65) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14345725 0.84 CYP1A1 (0.57) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14345762 0.81 CYP1A2 (0.63) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL4702182 0.81 CYP1A2 (0.62) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14345741 0.78 CYP1A2 (0.57) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL31402832 0.76 CYP1A1 (1.00) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14345924 0.75 CYP1A2 (0.63) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL4698728 0.73 CYP1A2 (0.66) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14345763 0.72 CYP1A2 (0.59) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL14346052 0.72 CYP1A1 (0.60) CYP1A2CYP1A1CYP1B1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007138081-A1 PYRIMIDINO[1',6'-1,2]PYRIDO[3,4-b]INDOLE DERIVATIVES AND THEIR THERAPEUTIC USAGE FOURTILLAN (FR) 2007-12-06 WO disclosed