SCHEMBL14347488

SCHEMBL14347488

CCOC(=O)c1cn(-c2cccc(-c3cccnc3)c2)c2ncccc2c1=O

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.65
PDE4A P27815 14/20 0.60
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
PDE4B Q07343 4/20 0.48
PDE4D Q08499 4/20 0.48
PDE4C Q08493 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7176953 0.90 KCNH2 (0.54) KCNH2PDE4ANPC1RAB9A
SCHEMBL5339663 0.89 PDE4A (0.76) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL8349787 0.86 KCNH2 (0.66) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL5342005 0.86 PDE4A (0.72) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL8247255 0.86 ELANE (0.58) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL8437043 0.84 PDE4A (0.54) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL1565419 0.84 PDE4A (0.70) KCNH2PDE4ANPC1RAB9A
SCHEMBL6135868 0.84 KCNH2 (0.71) KCNH2PDE4APDE4BPDE4DPDE4C
SCHEMBL7185413 0.84 PDE4A (0.65) KCNH2PDE4A
SCHEMBL7185969 0.83 PDE4A (0.62) KCNH2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312334-B2 Method of preparing inhibitors phosphodiesterase-4 MERCK & CO. INC. (US) 2007-12-25 US disclosed