SCHEMBL14367228

SCHEMBL14367228

O=C1Nc2ccccc2O[C@H](c2ccccc2)[C@@H]1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.56
HPGD P15428 2/20 0.51
HSD17B10 Q99714 2/20 0.51
USP2 O75604 2/20 0.51
THRB P10828 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ESR1 P03372 1/20 0.51
POLB P06746 1/20 0.51
ALOX15 P16050 1/20 0.51
PTPN7 P35236 1/20 0.51
RECQL P46063 1/20 0.51
ESR2 Q92731 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
RET P07949 1/20 0.44
KDR P35968 1/20 0.44
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903088 1.00 PARP1 (0.56) PARP1HPGDHSD17B10USP2THRB
SCHEMBL3346129 1.00 PARP1 (0.56) PARP1HPGDHSD17B10USP2THRB
SCHEMBL3344870 1.00 PARP1 (0.56) PARP1HPGDHSD17B10USP2THRB
SCHEMBL3342685 0.82 RET (0.48) PARP1HPGDHSD17B10USP2THRB
SCHEMBL3343396 0.82 PARP1 (0.54) PARP1HPGDHSD17B10USP2THRB
SCHEMBL4923583 0.82 PARP1 (0.54) PARP1HPGDHSD17B10USP2THRB
SCHEMBL13991180 0.82 PARP1 (0.54) PARP1HPGDHSD17B10USP2THRB
Hydrochloric Acid SCHEMBL4907950 0.81 PARP1 (0.53) PARP1HPGDHSD17B10USP2THRB
Hydrochloric Acid SCHEMBL4901800 0.81 PARP1 (0.53) PARP1HPGDHSD17B10USP2THRB
Hydrochloric Acid SCHEMBL4110963 0.81 PARP1 (0.53) PARP1HPGDHSD17B10USP2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294622-B2 Lactams and uses thereof ASTRAZENECA AB (SE) 2007-11-13 US disclosed
US-7294622-B2 Lactams and uses thereof ASTRAZENECA AB (SE) 2007-11-13 US disclosed