SCHEMBL14382004

SCHEMBL14382004

Oc1ccc2c(c1)CCN(c1ccc(F)cc1)C2Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.73
ESR2 Q92731 13/20 0.73
DRD2 P14416 2/20 0.46
DRD1 P21728 2/20 0.46
CYP26A1 O43174 1/20 0.44
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14381982 0.93 ESR1 (0.84) ESR1ESR2DRD2DRD1
SCHEMBL5103165 0.92 ESR1 (0.73) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL5108754 0.91 ESR1 (0.71) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL5664212 0.89 ESR1 (0.60) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL5524037 0.86 ESR1 (0.92) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL6716630 0.85 ESR1 (1.00) ESR1ESR2DRD2DRD1
SCHEMBL5641689 0.85 ESR1 (0.63) ESR1ESR2DRD2DRD1KDM4E
Hydrochloric Acid SCHEMBL5640529 0.84 ESR1 (0.61) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL5108599 0.83 ESR1 (0.60) ESR1ESR2DRD2DRD1KDM4E
SCHEMBL5105837 0.83 ESR1 (0.86) ESR1ESR2DRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279489-B2 Compounds and methods for modulation of estrogen receptors SIGNAL PHARMACEUTICALS, LLC (US) 2007-10-09 US disclosed