SCHEMBL14388166

SCHEMBL14388166

CNc1cc2ccn(-c3ccc(NC(=O)NS(=O)(=O)c4ccc(CI)s4)cn3)c(=O)c2cc1F

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 1/20 0.47
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
NOD1 Q9Y239 1/20 0.31
FBP1 P09467 1/20 0.30
TYK2 P29597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690441 0.90 P2RY12 (0.57) P2RY12CA12CA1CA2CA9
SCHEMBL14388167 0.89 P2RY12 (0.41) P2RY12NOD1FBP1
SCHEMBL14388082 0.88 P2RY12 (0.48) P2RY12CA12CA9NOD1
SCHEMBL14388093 0.86 P2RY12 (0.46) P2RY12CA12CA1CA2CA9
SCHEMBL14388193 0.86 P2RY12 (0.43) P2RY12NOD1FBP1
SCHEMBL14388192 0.85 P2RY12 (0.42) P2RY12NOD1FBP1
SCHEMBL14388169 0.85 P2RY12 (0.43) P2RY12NOD1TYK2
SCHEMBL14388191 0.84 P2RY12 (0.46) P2RY12NOD1
SCHEMBL14387887 0.83 P2RY12 (0.43) P2RY12CA12CA1CA2NOD1
SCHEMBL9922716 0.82 P2RY12 (0.48) P2RY12CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835444-B2 Cyclohexyl amide derivatives as CRF receptor antagonists NOVARTIS AG (CH) 2014-09-16 US disclosed
US-7294635-B2 Substituted isoquinolinones PORTOLA PHARMACEUTICALS, INC. (US) 2007-11-13 US disclosed