SCHEMBL14396830

SCHEMBL14396830

Nc1ccc(-c2cc(Oc3ccc4nc(NC5CCCCC5)sc4c3)ccn2)cn1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 15/20 0.60
PDGFRB P09619 4/20 0.54
KIT P10721 4/20 0.54
PDGFRA P16234 4/20 0.54
FLT3 P36888 4/20 0.54
ABL1 P00519 1/20 0.48
PIK3CA P42336 2/20 0.43
CYP3A4 P08684 1/20 0.43
NPC1 O15118 2/20 0.43
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14396835 0.91 CSF1R (0.59) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396649 0.89 CSF1R (0.54) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL2676949 0.88 CSF1R (0.64) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL19415479 0.88 CSF1R (0.52) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL2676384 0.87 CSF1R (0.45) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396988 0.87 CSF1R (0.52) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396996 0.87 CSF1R (0.52) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396834 0.86 CSF1R (0.65) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396486 0.86 CSF1R (0.59) CSF1RPDGFRBKITPDGFRAFLT3
SCHEMBL14396487 0.86 CSF1R (0.67) CSF1RPDGFRBKITPDGFRAFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010528-B1 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING NOVARTIS AG (CH) 2017-10-04 EP disclosed
WO-2007121484-A2 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING NOVARTIS AG (CH) 2007-10-25 WO disclosed