SCHEMBL14399400

SCHEMBL14399400

COc1cc(OC)c(Nc2nc(N)n(-c3cc(NC4CCCCC4)ncn3)n2)cc1CI

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 6/20 0.49
KIT P10721 5/20 0.49
IRAK4 Q9NWZ3 5/20 0.49
AURKA O14965 3/20 0.49
PDGFRB P09619 2/20 0.37
PDGFRA P16234 2/20 0.37
AXL P30530 6/20 0.36
JAK2 O60674 1/20 0.36
INSR P06213 4/20 0.36
KDR P35968 4/20 0.36
S1PR1 P21453 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAP4K1 Q92918 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
BACE1 P56817 1/20 0.34
TTK P33981 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12845487 0.88 FLT3 (0.49) FLT3KITIRAK4AURKAPDGFRB
SCHEMBL12779856 0.88 FLT3 (0.49) FLT3KITIRAK4AURKAPDGFRB
SCHEMBL12779908 0.86 FLT3 (0.64) FLT3KITIRAK4AURKAAXL
SCHEMBL12779850 0.85 KIT (0.52) FLT3KITIRAK4AURKAAXL
SCHEMBL13963811 0.83 FLT3 (0.47) FLT3KITIRAK4AURKAPDGFRB
SCHEMBL12779962 0.77 FLT3 (0.62) FLT3KITIRAK4AURKAAXL
SCHEMBL12779937 0.77 MEN1 (0.44) FLT3KITIRAK4AURKAPDGFRB
SCHEMBL12779942 0.75 KIT (0.59) FLT3KITIRAK4AURKAMEN1
SCHEMBL12779955 0.74 FLT3 (0.61) FLT3KITIRAK4AURKAAXL
SCHEMBL12779965 0.73 KIT (0.59) FLT3KITIRAK4AURKAAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279469-B2 Diaminotriazoles useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-09 US disclosed