SCHEMBL14411978

SCHEMBL14411978

CN(C)CC1CCCCN1c1n[nH]c2nccc(Cc3ccc(NC(=O)c4ccnn(-c5ccc(F)cc5)c4=O)cc3F)c12

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AXL P30530 20/20 0.54
MERTK Q12866 20/20 0.54
TYRO3 Q06418 15/20 0.54
MET P08581 19/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14411988 0.91 AXL (0.54) AXLMERTKTYRO3MET
SCHEMBL3109241 0.88 AXL (0.69) AXLMERTKTYRO3MET
SCHEMBL14412010 0.85 AXL (0.53) AXLMERTKTYRO3MET
SCHEMBL14411901 0.80 AXL (0.67) AXLMERTKTYRO3MET
SCHEMBL14411941 0.80 AXL (0.64) AXLMERTKTYRO3MET
SCHEMBL3109010 0.79 AXL (0.69) AXLMERTKTYRO3MET
SCHEMBL3109001 0.79 AXL (0.69) AXLMERTKTYRO3MET
SCHEMBL14411847 0.79 AXL (0.64) AXLMERTKTYRO3MET
SCHEMBL13905992 0.78 AXL (0.55) AXLMERTKTYRO3MET
SCHEMBL14411987 0.76 AXL (0.57) AXLMERTKTYRO3MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007103308-A2 HETEROBICYCLIC PYRAZOLE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-09-13 WO disclosed