SCHEMBL14419986

SCHEMBL14419986

O=Cc1ccc2c(c1)/C(=C/CCN1CCC(c3ccc(Cl)cc3)CC1)c1cccnc1CO2

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.55
CHRM2 P08172 1/20 0.55
CCR5 P51681 1/20 0.55
DRD2 P14416 2/20 0.36
DRD3 P35462 1/20 0.34
KCNH2 Q12809 1/20 0.34
CCR2 P41597 6/20 0.34
HRH1 P35367 3/20 0.34
ADRB2 P07550 1/20 0.34
ADRA2A P08913 1/20 0.34
CX3CR1 P49238 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14419987 0.89 CCR1 (0.53) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL14419953 0.89 CCR1 (0.56) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL12121935 0.88 CCR1 (0.52) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL13620898 0.87 CCR1 (0.71) CCR1CHRM2CCR5HRH1
SCHEMBL7212910 0.86 CCR1 (0.54) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL7212913 0.86 CCR1 (0.54) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL16312680 0.86 CCR1 (0.52) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL10288233 0.86 CCR1 (0.53) CCR1CHRM2CCR5DRD2DRD3
SCHEMBL14579629 0.85 CCR1 (0.62) CCR1CHRM2CCR5DRD2HRH1
SCHEMBL13620879 0.85 CCR1 (0.56) CCR1CHRM2CCR5DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271176-B2 Chemokine receptor antagonists and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-09-18 US disclosed