SCHEMBL14420177

SCHEMBL14420177

CC(C)N(Cc1ccc(Cl)cc1)[C@@H]1CCN(CC/C=C2/c3cc(C(C)(C)O)ccc3OCc3ncccc32)C1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.62
CHRM2 P08172 1/20 0.48
CCR5 P51681 1/20 0.48
HRH1 P35367 5/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
MCHR1 Q99705 1/20 0.32
TBXA2R P21731 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL656051 1.00 CCR1 (0.62) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL656050 1.00 CCR1 (0.62) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL652819 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL654801 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL10288003 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL653479 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL653480 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL15478339 0.91 CCR1 (0.60) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL656199 0.91 CCR1 (0.62) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL656198 0.91 CCR1 (0.62) CCR1CHRM2CCR5HRH1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8653096-B2 Chemokine receptor antagonists and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-02-18 US disclosed
US-7271176-B2 Chemokine receptor antagonists and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-09-18 US disclosed