SCHEMBL14423902

SCHEMBL14423902

NC(=O)c1cc2c(Oc3ccc(NC(=O)NC4CC4)c(Cl)c3)ccnc2cc1OC[C@H](O)CC1CCCC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 13/20 0.73
RET P07949 6/20 0.73
FGFR1 P11362 4/20 0.73
KDR P35968 3/20 0.73
PDGFRB P09619 3/20 0.73
PDGFRA P16234 3/20 0.73
FGFR2 P21802 3/20 0.73
FGFR3 P22607 3/20 0.73
KIT P10721 2/20 0.73
FLT1 P17948 2/20 0.73
FLT4 P35916 2/20 0.73
AURKB Q96GD4 2/20 0.73
RIPK2 O43353 1/20 0.73
ERN1 O75460 1/20 0.73
STK10 O94804 1/20 0.73
MAP3K6 O95382 1/20 0.73
ABL1 P00519 1/20 0.73
ESR1 P03372 1/20 0.73
ADORA3 P0DMS8 1/20 0.73
BCR P11274 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL863472 0.91 FGFR4 (0.77) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL863471 0.91 FGFR4 (0.77) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL1251009 0.89 FGFR4 (0.71) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL1251006 0.89 FGFR4 (0.71) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL1895467 0.87 FGFR4 (0.73) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL1895469 0.87 FGFR4 (0.73) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL1895420 0.87 FGFR4 (0.83) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL12412054 0.85 FGFR4 (0.79) FGFR4RETFGFR1KDRPDGFRB
SCHEMBL864110 0.85 FGFR4 (0.82) FGFR4RETFGFR1KDRPDGFRB
Lenvatinib SCHEMBL29372021 0.85 FGFR4 (1.00) FGFR4RETFGFR1KDRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253286-B2 Urea derivatives containing aromatic or heteroaromatic rings, useful as prophylactic or therapeutic agent for a disease for which angiogenesis inhibition is effective EISAI CO., LTD (JP) 2007-08-07 US disclosed
US-7253286-B2 Urea derivatives containing aromatic or heteroaromatic rings, useful as prophylactic or therapeutic agent for a disease for which angiogenesis inhibition is effective EISAI CO., LTD (JP) 2007-08-07 US disclosed