SCHEMBL14437495

SCHEMBL14437495

CN1CCN(c2ccc(NC(=O)c3cc(=O)c4cc(F)cc(N5CCN(C)CC5)c4[nH]3)cc2)CC1

nearest known ligand 0.91

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 8/20 0.91
SETD2 Q9BYW2 2/20 0.52
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
PLA2G7 Q13093 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
MAP4K4 O95819 1/20 0.46
LCK P06239 1/20 0.46
CYP3A4 P08684 1/20 0.46
CHRM1 P11229 1/20 0.46
CYP2C19 P33261 1/20 0.46
KDR P35968 1/20 0.46
TNIK Q9UKE5 1/20 0.46
RHEB Q15382 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14263970 0.95 HTR1B (1.00) HTR1BSETD2NPC1RAB9AMAPT
SCHEMBL14263971 0.92 HTR1B (0.78) HTR1BSETD2MAPTCYP2C19
SCHEMBL14437527 0.89 HTR1B (0.74) HTR1BSETD2NPC1RAB9APLA2G7
SCHEMBL14263965 0.84 HTR1B (1.00) HTR1BNPC1RAB9APLA2G7MAPT
SCHEMBL14437530 0.84 HTR1B (0.66) HTR1BSETD2RAB9APLA2G7MAPT
SCHEMBL14263964 0.81 HTR1B (0.79) HTR1BNPC1RAB9AMAPTHPGD
SCHEMBL5352760 0.81 HTR1B (1.00) HTR1BNPC1RAB9A
SCHEMBL4988305 0.81 HTR1B (0.61) HTR1B
Hydrochloric Acid SCHEMBL4982786 0.80 HTR1B (0.60) HTR1B
SCHEMBL14263955 0.78 HTR1B (0.77) HTR1BNPC1RAB9AMAP4K4TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007097697-A1 THERAPEUTIC QUINOLINE COMPOUNDS THAT ARE 5HT1B MODULATORS ASTRAZENECA AB (SE) 2007-08-30 WO disclosed