SCHEMBL14460641

SCHEMBL14460641

CC(=O)N1CCN(C(=O)c2cc(Sc3cnc(NC(=O)OC(C)(C)C)s3)ccc2O)CC1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITK Q08881 16/20 0.67
NTRK1 P04629 3/20 0.53
CDK2 P24941 1/20 0.51
TXK P42681 1/20 0.49
JAK3 P52333 1/20 0.49
BTK Q06187 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14460463 0.86 ITK (0.69) ITKNTRK1CDK2BTK
SCHEMBL14460626 0.84 ITK (0.80) ITK
SCHEMBL5656418 0.83 NTRK1 (0.46) ITKNTRK1CDK2
SCHEMBL5658013 0.80 ITK (1.00) ITK
SCHEMBL14461030 0.79 ITK (0.79) ITKNTRK1CDK2
SCHEMBL14460989 0.79 ITK (1.00) ITKNTRK1CDK2JAK3BTK
SCHEMBL14461032 0.78 ITK (0.77) ITKNTRK1CDK2
SCHEMBL14461031 0.78 ITK (1.00) ITKNTRK1CDK2
SCHEMBL14461038 0.78 ITK (0.73) ITKNTRK1CDK2
SCHEMBL14461000 0.77 ITK (0.83) ITKNTRK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7241781-B2 2-(pyridinylamino)thiazolylthio(optional methyl)-benzamides or -benzenealkanamides; may also contain antiinflammatory agents, antiproliferative agents, anticancer agents or anticytotoxic agents. BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-10 US disclosed
US-7241781-B2 2-(pyridinylamino)thiazolylthio(optional methyl)-benzamides or -benzenealkanamides; may also contain antiinflammatory agents, antiproliferative agents, anticancer agents or anticytotoxic agents. BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-10 US disclosed