SCHEMBL14508237

SCHEMBL14508237

CN(C)C1CCN(c2ccc(Nc3nc(N)c(C(=O)c4ccc(Cl)c(C#N)c4)s3)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 12/20 0.52
CCND1 P24385 12/20 0.52
CDK11A Q9UQ88 11/20 0.51
CCNT1 O60563 10/20 0.51
CDK9 P50750 10/20 0.51
CDK6 Q00534 10/20 0.51
CDK5 Q00535 4/20 0.51
GSK3A P49840 2/20 0.51
GSK3B P49841 2/20 0.51
LTK P29376 1/20 0.51
CLK2 P49760 1/20 0.51
CDK7 P50613 1/20 0.51
LIMK1 P53667 1/20 0.51
PRKCQ Q04759 1/20 0.51
TAOK1 Q7L7X3 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
ALK Q9UM73 1/20 0.51
CDK5R1 Q15078 3/20 0.46
TUBB8B A6NNZ2 1/20 0.44
TUBB4A P04350 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4338443 0.90 CDK4 (0.56) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4338779 0.87 GSK3A (0.65) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4333416 0.86 CDK4 (0.61) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4333581 0.86 CDK4 (0.58) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4331507 0.85 CDK4 (0.51) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4336041 0.84 CDK4 (0.56) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4337167 0.83 CDK4 (0.62) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4336279 0.83 CDK4 (0.62) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL13785057 0.83 CDK4 (0.61) CDK4CCND1CDK11ACCNT1CDK9
SCHEMBL4338041 0.83 CDK4 (0.61) CDK4CCND1CDK11ACCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7211576-B2 Diaminothiazoles HOFFMANN-LA ROCHE INC. (US) 2007-05-01 US disclosed
US-7211576-B2 Diaminothiazoles HOFFMANN-LA ROCHE INC. (US) 2007-05-01 US disclosed