SCHEMBL14517877

SCHEMBL14517877

O=C(O)C1CN(Cc2ccc(-c3noc(-c4ccc(C(F)(F)F)cc4)n3)cc2)C1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.81
S1PR5 Q9H228 16/20 0.81
S1PR4 O95977 13/20 0.81
S1PR3 Q99500 8/20 0.81
KCNH2 Q12809 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739441 0.89 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL3749519 0.88 S1PR1 (0.98) S1PR1S1PR5S1PR4S1PR3
SCHEMBL14517886 0.88 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL13415797 0.87 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL14517875 0.87 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL14517892 0.86 S1PR1 (0.89) S1PR1S1PR5S1PR4S1PR3
SCHEMBL15384213 0.86 S1PR1 (0.81) S1PR1S1PR5S1PR4S1PR3
SCHEMBL14517878 0.85 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3
SCHEMBL14176230 0.84 S1PR1 (0.73) S1PR1S1PR5S1PR4S1PR3
SCHEMBL13271364 0.84 S1PR1 (1.00) S1PR1S1PR5S1PR4S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7199142-B2 1-((5-aryl-1,2,4-oxadiazol-3-yl) benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl) pyrrolidine-3-carboxylates as edg receptor agonists MERCK & CO., INC. (US) 2007-04-03 US disclosed
US-7199142-B2 1-((5-aryl-1,2,4-oxadiazol-3-yl) benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl) pyrrolidine-3-carboxylates as edg receptor agonists MERCK & CO., INC. (US) 2007-04-03 US disclosed