SCHEMBL14520587

SCHEMBL14520587

C=Cc1nc(Nc2cc(C)[nH]n2)cc2cc(O)c(F)cc12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 6/20 0.38
JAK3 P52333 6/20 0.38
PLK4 O00444 3/20 0.37
NTRK1 P04629 9/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C8 P10632 3/20 0.36
CYP2C9 P11712 3/20 0.36
JAK1 P23458 3/20 0.36
TYK2 P29597 3/20 0.36
CYP2C19 P33261 3/20 0.36
ADORA3 P0DMS8 2/20 0.36
CYP1A2 P05177 1/20 0.36
TNIK Q9UKE5 1/20 0.36
PAK4 O96013 1/20 0.35
NTRK3 Q16288 1/20 0.35
NTRK2 Q16620 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973293 0.82 JAK2 (0.39) JAK2JAK3PLK4NTRK1CYP3A4
SCHEMBL3966806 0.77 JAK2 (0.41) JAK2JAK3PLK4NTRK1CYP3A4
SCHEMBL3972231 0.71 AURKA (0.41) JAK2JAK3NTRK1CYP3A4NTRK3
SCHEMBL3967892 0.66 JAK2 (0.41) JAK2JAK3PLK4NTRK1JAK1
SCHEMBL3964062 0.65 NTRK1 (0.45) JAK2JAK3PLK4NTRK1CYP2C19
SCHEMBL3972216 0.64 SYK (0.46) PLK4NTRK1TNIKPAK4
SCHEMBL3972285 0.64 CCNA2 (0.45) PLK4NTRK1PAK4
SCHEMBL3969898 0.64 SYK (0.43) PLK4TNIKPAK4
SCHEMBL3969123 0.63 JAK2 (0.40) JAK2JAK3PLK4NTRK1JAK1
SCHEMBL3972230 0.63 AURKA (0.38) JAK2JAK3PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007071348-A1 ISOQUINOLINE AMINOPYRAZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2007-06-28 WO disclosed