SCHEMBL14526953

SCHEMBL14526953

Cc1cc(CC(NC(=O)N2CCC(N3CCc4ccccc4NC3=O)CC2)C(=O)N2CCC(N3CCNCC3)CC2)cc2cc[nH]c12

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.64
CYP3A4 P08684 16/20 0.64
RAMP1 O60894 2/20 0.54
CYP2D6 P10635 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14526959 0.96 CALCRL (0.62) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526945 0.94 CALCRL (0.60) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526946 0.94 CALCRL (0.64) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526957 0.93 CALCRL (0.64) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526944 0.91 CALCRL (0.61) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526787 0.90 CALCRL (0.79) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526937 0.89 CALCRL (0.62) CALCRLCYP3A4
SCHEMBL14526791 0.88 CALCRL (0.79) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL14526925 0.87 CALCRL (0.63) CALCRLCYP3A4RAMP1CYP2D6
SCHEMBL5660798 0.87 CALCRL (0.63) CALCRLCYP3A4RAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205294-B2 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-04-17 US disclosed
US-7205294-B2 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-04-17 US disclosed