SCHEMBL14535372

SCHEMBL14535372

COc1ccc([C@H](O)CNC2CNC(=O)C2c2nc3c(C)cc(N4CCOCC4)cc3[nH]2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 19/20 0.47
CYP3A4 P08684 16/20 0.47
PTK2 Q05397 3/20 0.47
EGFR P00533 2/20 0.47
INSR P06213 2/20 0.47
LCK P06239 2/20 0.47
KDR P35968 2/20 0.47
AURKA O14965 2/20 0.47
AURKB Q96GD4 2/20 0.47
ALK Q9UM73 2/20 0.47
ERBB2 P04626 1/20 0.47
CYP1A2 P05177 1/20 0.47
MET P08581 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAP2K1 Q02750 1/20 0.47
PLK4 O00444 1/20 0.47
CHEK1 O14757 1/20 0.47
PDPK1 O15530 1/20 0.47
DAPK3 O43293 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14535394 0.87 IGF1R (0.61) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL5509849 0.79 IGF1R (0.55) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL14510495 0.79 IGF1R (0.55) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL4136625 0.77 IGF1R (0.78) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL5138375 0.77 IGF1R (0.78) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL14535409 0.74 IGF1R (0.60) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL4426826 0.71 IGF1R (0.69) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL14510464 0.71 IGF1R (0.69) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL5137354 0.71 IGF1R (0.69) IGF1RCYP3A4PTK2EGFRINSR
SCHEMBL5137353 0.71 IGF1R (0.69) IGF1RCYP3A4PTK2EGFRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7223757-B2 Tyrosine kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-29 US disclosed