SCHEMBL14540802

SCHEMBL14540802

O=c1[nH]nc2c(-c3ccc(Cl)cc3)c(-c3ccc(Cl)cc3)c3nn(Cc4ccc(C(F)(F)F)cc4)c(=O)n3n12

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 17/20 0.54
CYP3A4 P08684 4/20 0.47
CYP2C9 P11712 4/20 0.47
CYP2C19 P33261 4/20 0.47
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
P2RX3 P56373 1/20 0.40
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14540419 0.86 CNR1 (0.75) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL13135224 0.86 CNR1 (0.51) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL3550472 0.82 CNR1 (0.51) CNR1CYP3A4CYP2C9CYP2C19P2RX3
SCHEMBL13114629 0.82 CNR1 (0.75) CNR1CYP3A4CYP2C9CYP2C19NR1H2
SCHEMBL14540568 0.82 CNR1 (0.72) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL14540423 0.82 CNR1 (0.56) CNR1CYP3A4CYP2C9CYP2C19NR1H2
SCHEMBL14540421 0.81 CNR1 (0.60) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL14540718 0.80 CNR1 (0.54) CNR1CYP3A4CYP2C9CYP2C19NR1H2
SCHEMBL13114630 0.80 CNR1 (0.65) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL13114639 0.78 CNR1 (0.73) CNR1CYP3A4CYP2C9CYP2C19NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697371-B1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-04-25 EP disclosed