SCHEMBL14540933

SCHEMBL14540933

N#Cc1cc2c(Oc3ccc(NC(=O)NC4CC4)c(F)c3)ccnc2cc1OCCCCO

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 8/20 0.53
KDR P35968 8/20 0.50
PDGFRA P16234 5/20 0.50
KIT P10721 4/20 0.50
FGFR2 P21802 4/20 0.50
AXL P30530 3/20 0.50
FGFR1 P11362 3/20 0.49
FGFR3 P22607 3/20 0.49
RET P07949 3/20 0.49
RIPK2 O43353 1/20 0.49
ERN1 O75460 1/20 0.49
STK10 O94804 1/20 0.49
MAP3K6 O95382 1/20 0.49
ABL1 P00519 1/20 0.49
ESR1 P03372 1/20 0.49
PDGFRB P09619 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
BCR P11274 1/20 0.49
NQO2 P16083 1/20 0.49
FLT1 P17948 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1249397 0.91 FGFR4 (0.57) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL14540600 0.89 KDR (0.56) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL13627606 0.88 FGFR4 (0.52) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1894739 0.88 KDR (0.55) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1891355 0.88 FGFR4 (0.55) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1891352 0.88 FGFR4 (0.55) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1893066 0.86 FGFR4 (0.52) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1895735 0.85 FGFR4 (0.56) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1890074 0.85 KDR (0.53) FGFR4KDRPDGFRAKITFGFR2
SCHEMBL1896810 0.84 FGFR4 (0.57) FGFR4KDRPDGFRAKITFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1777218-A1 Process for the preparation of 4-phenoxy quinoline derivatives Eisai R&D Management Co., Ltd. (JP) 2007-04-25 EP disclosed