SCHEMBL14541014

SCHEMBL14541014

N#Cc1ccc(Cn2nc3c(-c4ccc(Cl)cc4)c(-c4ccc(Cl)cc4)cnn3c2=O)nc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.53
CYP3A4 P08684 1/20 0.45
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
RIPK3 Q9Y572 1/20 0.36
P2RX3 P56373 1/20 0.35
MDM2 Q00987 1/20 0.35
NT5E P21589 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP11B2 P19099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14181001 0.95 CNR1 (0.60) CNR1CYP3A4RIPK3CYP2C19
SCHEMBL4802818 0.88 CNR1 (0.61) CNR1CYP3A4KDM4EALDH1A1LMNA
SCHEMBL4803698 0.83 CNR1 (0.69) CNR1CYP3A4RIPK3CYP2C19CYP11B2
SCHEMBL14180936 0.83 CNR1 (0.57) CNR1CYP3A4KDM4EALDH1A1LMNA
SCHEMBL4805900 0.82 CNR1 (0.62) CNR1CYP3A4LMNACYP2C19
SCHEMBL14180898 0.82 CNR1 (0.58) CNR1CYP3A4KDM4EALDH1A1LMNA
SCHEMBL14180933 0.82 CNR1 (0.64) CNR1CYP3A4KDM4ECYP2C19
SCHEMBL14180823 0.82 CNR1 (0.54) CNR1CYP3A4KDM4E
SCHEMBL14181064 0.81 CNR1 (0.66) CNR1CYP3A4CYP2C19
SCHEMBL4800125 0.81 CNR1 (0.70) CNR1CYP3A4KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697370-B1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-04-25 EP disclosed