SCHEMBL14547856

SCHEMBL14547856

CC(C)NC(=O)c1ccc(Nc2nc(NCC(F)(F)F)c3cc[nH]c3n2)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 6/20 0.58
PTK2 Q05397 12/20 0.58
ROCK1 Q13464 6/20 0.58
JAK2 O60674 6/20 0.58
RET P07949 6/20 0.58
MAPK8 P45983 6/20 0.58
MAP4K2 Q12851 6/20 0.58
NTRK2 Q16620 5/20 0.58
AURKA O14965 5/20 0.58
PAK4 O96013 5/20 0.58
LTK P29376 5/20 0.58
KDR P35968 5/20 0.58
MAPK9 P45984 5/20 0.58
RPS6KA3 P51812 5/20 0.58
JAK3 P52333 5/20 0.58
MAP2K1 Q02750 5/20 0.58
MST1R Q04912 5/20 0.58
AURKB Q96GD4 5/20 0.58
CLK4 Q9HAZ1 5/20 0.58
ALK Q9UM73 5/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14547851 0.90 LRRK2 (0.59) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547718 0.90 LRRK2 (0.61) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547719 0.90 PTK2 (0.59) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547857 0.89 PTK2 (0.64) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547943 0.87 PTK2 (0.60) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547767 0.87 PTK2 (0.75) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14287397 0.85 PTK2 (0.75) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547785 0.83 LRRK2 (0.58) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547974 0.81 LRRK2 (0.55) LRRK2PTK2ROCK1JAK2RET
SCHEMBL14547771 0.81 LRRK2 (0.57) LRRK2PTK2ROCK1JAK2RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007042299-A1 PYRROLOPYRIMIDINE DERIVATIVES AS SYK INHIBITORS GLAXO GROUP LIMITED (GB) 2007-04-19 WO disclosed