SCHEMBL14548958

SCHEMBL14548958

NCCNC(=O)Cn1cnc2c(NC(=O)OCc3ccccc3)ncnc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.55
HDAC2 Q92769 8/20 0.55
TDP1 Q9NUW8 2/20 0.47
HTT P42858 1/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA9 Q16790 2/20 0.44
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
TMIGD3 P0DMS9 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
ADORA2B P29275 1/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
EGFR P00533 1/20 0.41
DOT1L Q8TEK3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3130095 0.86 TDP1 (0.48) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL7906492 0.84 PDE4A (0.49) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL8421549 0.82 PDE4A (0.47) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL6690200 0.82 TDP1 (0.49) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL6803674 0.81 HDAC1 (0.46) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL14548981 0.80 MEN1 (0.42) HDAC1HDAC2HDAC8HDAC6
SCHEMBL9435466 0.80 CCNE2 (0.47) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL13609069 0.79 HTT (0.57) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL13196022 0.78 NPC1 (0.45) HDAC1HDAC2TDP1HTTPDE4A
SCHEMBL11986874 0.78 CDK1 (0.59) PDE4APDE4BPDE4CPDE4DTMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189941-B1 NEUROMEDIN B AND SOMATOSTATIN RECEPTOR AGONISTS IPSEN PHARMA (FR) 2013-01-09 EP disclosed