SCHEMBL14567705

SCHEMBL14567705

Bc1c(Cn2nc(-c3ccccc3)c3c(Cl)nc(N)nc32)nc(OC)c(OC)c1C

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.46
TRAP1 Q12931 2/20 0.39
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
RICTOR Q6R327 1/20 0.38
RPTOR Q8N122 1/20 0.38
MAPKAP1 Q9BPZ7 1/20 0.38
MLST8 Q9BVC4 1/20 0.38
HSP90AB1 P08238 3/20 0.36
FYN P06241 1/20 0.35
HSP90B1 P14625 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3424934 0.81 HSP90AA1 (0.68) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14506500 0.76 HSP90AA1 (0.57) HSP90AA1TRAP1PIK3CAMTORRICTOR
SCHEMBL3391504 0.75 HSP90AA1 (0.54) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL3393039 0.74 HSP90AA1 (0.54) HSP90AA1TRAP1PIK3CAMTORRICTOR
SCHEMBL14506471 0.71 HSP90AA1 (0.41) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14506499 0.69 HSP90AA1 (0.42) HSP90AA1PIK3CAMTORRICTORRPTOR
SCHEMBL8129925 0.66 PIK3CD (0.50) PIK3CA
SCHEMBL3393936 0.66 HSP90AA1 (0.69) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL3396133 0.64 HSP90AA1 (0.66) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14568048 0.64 HSP90AA1 (0.49) HSP90AA1TRAP1HSP90AB1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007035963-A2 ANTI-TUMOR METHODS USING MULTI DRUG RESISTANCE INDEPENDENT SYNTHETIC HSP90 INHIBITORS CONFORMA THERAPEUTICS CORPORATION (US) 2007-03-29 WO disclosed