SCHEMBL14568043

SCHEMBL14568043

COc1nc(Cn2ncc3c(Cl)nc(N)nc32)c(Br)c(OC)c1OC

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.62
TRAP1 Q12931 5/20 0.62
HSP90AB1 P08238 12/20 0.48
HSP90B1 P14625 2/20 0.47
ADA P00813 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14506465 0.89 HSP90AA1 (0.65) HSP90AA1TRAP1HSP90AB1HSP90B1ADA
SCHEMBL13539431 0.86 HSP90AA1 (0.61) HSP90AA1TRAP1HSP90AB1HSP90B1ADA
SCHEMBL14568309 0.83 HSP90AA1 (0.73) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL13539434 0.80 HSP90AA1 (0.61) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14568308 0.80 HSP90AA1 (0.72) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14568297 0.80 HSP90AA1 (0.63) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14567904 0.79 HSP90AA1 (0.44) HSP90AA1TRAP1HSP90AB1HSP90B1ADORA2A
SCHEMBL3397593 0.79 HSP90AA1 (0.76) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL14568045 0.78 HSP90AA1 (0.71) HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL3390492 0.77 HSP90AA1 (1.00) HSP90AA1TRAP1HSP90AB1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007035963-A2 ANTI-TUMOR METHODS USING MULTI DRUG RESISTANCE INDEPENDENT SYNTHETIC HSP90 INHIBITORS CONFORMA THERAPEUTICS CORPORATION (US) 2007-03-29 WO disclosed