SCHEMBL14568280

SCHEMBL14568280

COc1cc(Cn2cnc3c(C)nc(N)nc32)nc(OC)c1OC

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 18/20 0.67
HSP90AA1 P07900 17/20 0.67
HSP90B1 P14625 1/20 0.45
TRAP1 Q12931 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14438223 0.88 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3389635 0.80 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3393558 0.77 HSP90AB1 (0.77) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL14568282 0.74 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3395258 0.73 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3394915 0.73 HSP90AA1 (0.78) HSP90AB1HSP90AA1
SCHEMBL14568279 0.73 HSP90AA1 (0.80) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3394034 0.71 HSP90AB1 (0.76) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3393012 0.71 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL14438216 0.70 HSP90AB1 (0.67) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007035963-A2 ANTI-TUMOR METHODS USING MULTI DRUG RESISTANCE INDEPENDENT SYNTHETIC HSP90 INHIBITORS CONFORMA THERAPEUTICS CORPORATION (US) 2007-03-29 WO disclosed