SCHEMBL14570643

SCHEMBL14570643

Cn1cncc1C(O)(c1ccc2c(c1)c(-c1cccc(Cl)c1)cc1nnnn12)c1cc2ccccc2s1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 16/20 0.67
FNTB P49356 16/20 0.67
PGGT1B P53609 3/20 0.67
RORC P51449 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5016840 0.90 FNTA (0.78) FNTAFNTBPGGT1B
SCHEMBL5023612 0.89 FNTA (0.70) FNTAFNTBPGGT1BRORC
SCHEMBL5025653 0.88 FNTA (0.69) FNTAFNTBPGGT1BRORC
SCHEMBL6303247 0.87 FNTA (0.79) FNTAFNTBPGGT1BRORC
SCHEMBL14570645 0.87 FNTA (0.68) FNTAFNTBPGGT1BRORC
SCHEMBL3502124 0.85 FNTA (0.75) FNTAFNTBPGGT1B
SCHEMBL14570640 0.85 FNTA (0.64) FNTAFNTBPGGT1BRORC
SCHEMBL5023704 0.84 FNTA (0.69) FNTAFNTBPGGT1BRORC
SCHEMBL5023789 0.83 FNTA (0.68) FNTAFNTBPGGT1BRORC
SCHEMBL14570642 0.82 FNTA (0.67) FNTAFNTBPGGT1BRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196094-B2 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-27 US disclosed
US-7196094-B2 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-27 US disclosed