SCHEMBL14600256

SCHEMBL14600256

CCCc1nn(-c2ncccc2C)c(Nc2ccc(C3CC3)cc2C(=O)O)c1-c1ccc(OC)nc1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 8/20 0.44
ADORA1 P30542 12/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600253 0.90 DHODH (0.46) DHODHADORA1
SCHEMBL14600254 0.90 ADORA1 (0.51) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600455 0.89 DHODH (0.47) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600234 0.87 ADORA1 (0.51) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL4668599 0.84 ADORA1 (0.50) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600714 0.83 DHODH (0.42) DHODHADORA1ADORA2AADORA2B
SCHEMBL4668512 0.83 ADORA1 (0.41) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600994 0.82 ADORA1 (0.46) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600704 0.79 ADORA1 (0.46) DHODHADORA1ADORA3ADORA2AADORA2B
SCHEMBL14600257 0.79 DHODH (0.50) DHODHADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed