SCHEMBL14600655

SCHEMBL14600655

C=C(O)c1cc(OC(F)(F)F)ccc1Nc1c(-c2cccnc2F)c(CC)nn1-c1cccnc1C

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 17/20 0.41
ADORA3 P0DMS8 1/20 0.37
P2RY1 P47900 1/20 0.36
ADORA2B P29275 2/20 0.34
ADORA2A P29274 1/20 0.34
CCR9 P51686 1/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600659 0.91 ADORA1 (0.43) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL14600658 0.89 ADORA1 (0.43) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL14600656 0.87 ADORA1 (0.43) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL14600201 0.87 ADORA1 (0.42) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL14600657 0.87 ADORA1 (0.41) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL14600202 0.85 ADORA1 (0.45) ADORA1ADORA3ADORA2BADORA2A
SCHEMBL4666639 0.84 ADORA1 (0.50) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL4666620 0.81 ADORA1 (0.50) ADORA1ADORA3P2RY1ADORA2BADORA2A
SCHEMBL4669467 0.80 ADORA1 (0.49) ADORA1ADORA3ADORA2BADORA2ATP53
SCHEMBL4666643 0.80 ADORA1 (0.49) ADORA1ADORA3ADORA2BADORA2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed