SCHEMBL1460098

SCHEMBL1460098

O=C(ONC1CCCC1)C1=CN(C(=O)c2ccc(F)cc2)CCc2c1[nH]c1ccccc21

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 10/20 0.68
ABCB1 P08183 2/20 0.45
ABCG2 Q9UNQ0 2/20 0.45
CDK4 P11802 1/20 0.44
CCND1 P24385 1/20 0.44
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
ATM Q13315 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TRPV1 Q8NER1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL274621 0.88 NR1H4 (0.73) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL273780 0.87 NR1H4 (0.72) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL275327 0.86 NR1H4 (0.63) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL275994 0.86 NR1H4 (0.73) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL273104 0.86 NR1H4 (0.62) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL274682 0.85 NR1H4 (0.80) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL275053 0.85 NR1H4 (0.63) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL275227 0.83 NR1H4 (0.65) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL687653 0.82 NR1H4 (0.56) NR1H4ABCB1ABCG2CDK4CCND1
SCHEMBL275399 0.82 NR1H4 (0.75) NR1H4ABCB1ABCG2CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4646293-B2 2011-03-09 JP claimed
JP-2005531585-A 2005-10-20 JP claimed
EP-1532153-A1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X-Ceptor Therapeutics, Inc. (US) 2005-05-25 EP claimed
WO-2003099821-A1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X-CEPTOR THERAPEUTICS, INC. (US) 2003-12-04 WO claimed