SCHEMBL14601451

SCHEMBL14601451

O=C(O)c1ccc(N(CCC2CCCCC2)c2nc(-c3nc4cc(OCc5ccc(Cl)c(Cl)c5)ccc4[nH]3)cs2)cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.37
GCGR P47871 3/20 0.36
GIPR P48546 3/20 0.36
PRSS12 P56730 2/20 0.35
S1PR1 P21453 3/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
MDM2 Q00987 3/20 0.34
MDH2 P40926 1/20 0.33
CYP2D6 P10635 1/20 0.33
RXRB P28702 2/20 0.33
NPC1 O15118 1/20 0.33
RXRA P19793 1/20 0.33
RXRG P48443 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5585741 0.99 CHEK2 (0.37) CHEK2GCGRGIPRPRSS12S1PR1
Hydrochloric Acid SCHEMBL5585747 0.94 CHEK2 (0.42) CHEK2GCGRGIPRPRSS12MRGPRX4
SCHEMBL5585511 0.85 MAOB (0.41) GCGRGIPRS1PR1MRGPRX4CYP2D6
SCHEMBL5585453 0.81 MRGPRX4 (0.40) GCGRGIPRMRGPRX4NPC1RAB9A
SCHEMBL5585550 0.78 MAOB (0.41) GCGRGIPRMRGPRX4MDH2CYP2D6
SCHEMBL14601452 0.76 CSNK2A1 (0.45) MRGPRX4MDH2NPC1RAB9A
Hydrochloric Acid SCHEMBL5585667 0.76 CSNK2A1 (0.44) PRSS12MRGPRX4MDH2NPC1RAB9A
SCHEMBL5585545 0.74 HRH3 (0.43) GCGRGIPRS1PR1NPC1RAB9A
SCHEMBL5585721 0.73 KMT2A (0.46) GCGRGIPRMRGPRX4NPC1RAB9A
SCHEMBL5585777 0.72 PTGER1 (0.49) MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7163952-B2 Azole compound and medicinal use thereof JAPAN TOBACCO INC. (JP) 2007-01-16 US disclosed