SCHEMBL14604241

SCHEMBL14604241

COC(=O)c1[nH]c2c(-c3ccccc3)c(OC)ccc2c(=O)c1CNC(=O)c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 4/20 0.51
MAPT P10636 1/20 0.42
MAPK1 P28482 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 2/20 0.41
USP2 O75604 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.41
AAK1 Q2M2I8 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.40
BLM P54132 1/20 0.40
APLNR P35414 1/20 0.40
POLB P06746 1/20 0.40
CYP2C19 P33261 1/20 0.40
GALR3 O60755 1/20 0.40
NR2F2 P24468 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14604142 0.90 MAPK8 (0.53) MAPK8ALDH1A1KDM4ETSHRMEN1
SCHEMBL14604214 0.86 MAPK8 (0.51) MAPK8ALDH1A1MEN1KMT2A
SCHEMBL14604171 0.85 MAPK8 (0.53) MAPK8MAPTALDH1A1USP2TSHR
SCHEMBL14603845 0.85 MAPK8 (0.50) MAPK8
SCHEMBL14604205 0.85 MAPK8 (0.49) MAPK8
SCHEMBL14603998 0.85 MAPK8 (0.53) MAPK8
SCHEMBL14604394 0.84 MAPK8 (0.51) MAPK8KMT2A
SCHEMBL14604167 0.83 MAPK8 (0.52) MAPK8MEN1KMT2A
SCHEMBL14604008 0.80 MAPK8 (0.48) MAPK8
SCHEMBL14604039 0.80 MAPK8 (0.51) MAPK8MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2731932-A1 AMINOMETHYL QUINOLONE COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2014-05-21 EP disclosed
WO-2013007676-A1 AMINOMETHYL QUINOLONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2013-01-17 WO disclosed