SCHEMBL14604245

SCHEMBL14604245

CN(C)C(=O)c1[nH]c2c(-c3ccccc3)c(Cl)ccc2c(=O)c1CNC(=O)c1ccc2ncsc2c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 12/20 0.60
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
POLB P06746 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14604163 0.85 MAPK8 (0.58) MAPK8
SCHEMBL14604023 0.82 MAPK8 (0.53) MAPK8NPC1RAB9A
SCHEMBL14604348 0.77 MAPK8 (0.61) MAPK8
SCHEMBL14604228 0.76 MAPK8 (0.54) MAPK8
SCHEMBL14604334 0.75 GRIN1 (0.57) MAPK8MEN1KMT2A
SCHEMBL14576222 0.75 MAPK8 (1.00) MAPK8
SCHEMBL14604229 0.74 MAPK8 (0.49) MAPK8
SCHEMBL14604008 0.74 MAPK8 (0.48) MAPK8
SCHEMBL14604063 0.74 MAPK8 (0.56) MAPK8
SCHEMBL14604343 0.74 MAPK8 (0.55) MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2731932-A1 AMINOMETHYL QUINOLONE COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2014-05-21 EP disclosed
WO-2013007676-A1 AMINOMETHYL QUINOLONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2013-01-17 WO disclosed