SCHEMBL14607606

SCHEMBL14607606

CN(c1c2c(c(OC(c3ccccc3)c3ccccc3)c3ncccc13)C(=O)N(Cc1ccc(F)cc1)C2)S(=O)(=O)CCCC#N

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.32
PTGER4 P35408 5/20 0.31
AGTR2 P50052 1/20 0.31
CACNA2D1 P54289 1/20 0.31
KAT2B Q92831 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14573781 0.94 PTGER4 (0.33) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL14573780 0.92 TDP1 (0.33) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL14607607 0.92 IDH1 (0.32) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL12378082 0.91 IDH1 (0.34) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL14573777 0.89 IDH1 (0.34) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL14573782 0.89 HTT (0.36) CACNA2D1
SCHEMBL14573778 0.89 IDH1 (0.34) IDH1PTGER4CACNA2D1KAT2B
SCHEMBL12378100 0.88 PTGDR2 (0.32) IDH1PTGER4CACNA2D1
SCHEMBL12378101 0.86 IDH1 (0.33) IDH1PTGER4CACNA2D1
SCHEMBL12378113 0.86 TP53 (0.35) IDH1PTGER4CACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070072831-A1 Integrase inhibitor compounds GILEAD SCIENCES, INC. 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072831-A1 Integrase inhibitor compounds TYMP, CDKN1A, PAICS IDH1 104/4885PTGER4 3914/4885AGTR2 4618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.