SCHEMBL14625528

SCHEMBL14625528

CCC(=O)Nc1cccc(C2(c3cc(C(=O)CC)n(CC)c3)N=C(N)NC2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.41
KCNH2 Q12809 1/20 0.41
BACE2 Q9Y5Z0 3/20 0.39
RAB9A P51151 2/20 0.37
POLB P06746 1/20 0.37
NR4A1 P22736 1/20 0.37
GAA P10253 2/20 0.37
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
TP53 P04637 2/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14625674 0.95 BACE1 (0.44) BACE1KCNH2BACE2POLBGAA
SCHEMBL3580248 0.84 BACE1 (0.47) BACE1BACE2
SCHEMBL3572542 0.80 BACE1 (0.55) BACE1BACE2
SCHEMBL3579229 0.78 BACE1 (0.55) BACE1BACE2
SCHEMBL3588109 0.72 BACE1 (0.47) BACE1BACE2HPGDSMN1; SMN2
SCHEMBL14625360 0.71 BACE1 (0.53) BACE1BACE2
SCHEMBL7886785 0.70 BACE1 (0.49) BACE1BACE2
SCHEMBL3575427 0.70 BACE1 (0.49) BACE1BACE2
SCHEMBL7888135 0.69 BACE1 (0.63) BACE1BACE2
SCHEMBL3581817 0.69 BACE1 (0.52) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007005366-A1 AMlNO-5-(5-MEMBERED)HETEROARYLIMIDAZOLONE COMPOUNDS AND THE USE THEREOF FOR β-SECRETASE MODULATION WYETH (US) 2007-01-11 WO disclosed