SCHEMBL14636899

SCHEMBL14636899

CC1(C(=O)N2CCCC(C3=C4C=NC=C[N+]4(N)C(c4ccc(C(=O)Nc5cccnn5)cc4)=N3)C2)COC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.56
LCK P06239 1/20 0.41
LYN P07948 1/20 0.41
TEC P42680 1/20 0.41
TXK P42681 1/20 0.41
FRK P42685 1/20 0.41
BLK P51451 1/20 0.41
BMX P51813 1/20 0.41
KCNH2 Q12809 1/20 0.41
PTK6 Q13882 1/20 0.41
ERBB4 Q15303 1/20 0.41
SRMS Q9H3Y6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15914192 1.00 BTK (0.56) BTKLCKLYNTECTXK
SCHEMBL14631267 0.88 BTK (0.57) BTKLCKLYNTECTXK
SCHEMBL14630604 0.88 BTK (0.56) BTKLCKLYNTECTXK
SCHEMBL14637061 0.87 BTK (0.50) BTKLCKLYNTECTXK
SCHEMBL14636296 0.87 BTK (0.49) BTKLCKLYNTECTXK
SCHEMBL15913687 0.87 BTK (0.55) BTKLCKLYNTECTXK
SCHEMBL14636741 0.87 BTK (0.57) BTKLCKLYNTECTXK
SCHEMBL14636791 0.87 BTK (0.56) BTKLCKLYNTECTXK
SCHEMBL15913905 0.87 BTK (0.49) BTKLCKLYNTECTXK
SCHEMBL14637496 0.87 BTK (0.49) BTKLCKLYNTECTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2734529-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2014-05-28 EP disclosed
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed