SCHEMBL14637338

SCHEMBL14637338

COc1cc(C(=O)Nc2cc(C(F)(F)F)ccn2)ccc1C1=NC(C2CCCN(C(=O)C3(C)COC3)C2)=C2C=NC=C[N+]12N

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.61
LCK P06239 2/20 0.54
LYN P07948 2/20 0.54
TEC P42680 2/20 0.54
TXK P42681 2/20 0.54
FRK P42685 2/20 0.54
BLK P51451 2/20 0.54
BMX P51813 2/20 0.54
PTK6 Q13882 2/20 0.54
ERBB4 Q15303 2/20 0.54
SRMS Q9H3Y6 2/20 0.54
FYN P06241 1/20 0.54
YES1 P07947 1/20 0.54
FGR P09769 1/20 0.54
SRC P12931 1/20 0.54
CSK P41240 1/20 0.54
ITK Q08881 1/20 0.54
KCNH2 Q12809 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14636563 1.00 BTK (0.61) BTKLCKLYNTECTXK
SCHEMBL14636818 0.93 BTK (0.61) BTKLCKLYNTECTXK
SCHEMBL14637083 0.93 BTK (0.61) BTKLCKLYNTECTXK
SCHEMBL14636973 0.93 BTK (0.61) BTKLCKLYNTECTXK
SCHEMBL15913716 0.93 BTK (0.61) BTKLCKLYNTECTXK
SCHEMBL14637085 0.91 BTK (0.54) BTKLCKLYNTECTXK
SCHEMBL14630171 0.90 BTK (0.59) BTKLCKLYNTECTXK
SCHEMBL14636996 0.90 BTK (0.59) BTKLCKLYNTECTXK
SCHEMBL15913869 0.90 BTK (0.52) BTKLCKLYNTECTXK
SCHEMBL14638594 0.89 BTK (0.56) BTKLCKLYNTECTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed