SCHEMBL14643204

SCHEMBL14643204

CCCCC1(c2cncc(Br)c2)NC(=N)N(Cc2ccc(CNC(=O)NCCC)cc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.40
BACE1 P56817 6/20 0.40
USP2 O75604 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512910 0.97 BACE1 (0.43) HDAC6BACE1RXFP1SMN1; SMN2GAA
SCHEMBL7518509 0.84 HDAC6 (0.47) HDAC6BACE1RXFP1KMT2A
SCHEMBL7536228 0.84 BACE1 (0.44) HDAC6BACE1GAA
SCHEMBL7510758 0.81 HDAC6 (0.53) HDAC6BACE1
SCHEMBL17715612 0.79 RXFP1 (0.47) HDAC6RXFP1KMT2A
SCHEMBL11932498 0.79 HDAC6 (0.51) HDAC6BACE1RXFP1KMT2A
SCHEMBL13723059 0.79 HDAC6 (0.44) HDAC6BACE1RXFP1
SCHEMBL7519450 0.76 CNR1 (0.36)
SCHEMBL7513638 0.75 BACE1 (0.54) HDAC6BACE1RXFP1KMT2A
SCHEMBL7514490 0.75 BACE1 (0.50) HDAC6BACE1USP2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8778980-B2 Heterocyclic aspartyl protease inhibitors MERCK SHARP & DOHME CORP. (US) 2014-07-15 US disclosed
US-20130018066-A1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS Schering Corporation & Pharmacopeia Drug Discovery Inc. (US) 2013-01-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130018066-A1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS CHRM1, CHRM2, PRSS1 HDAC6 2138/4885BACE1 8/4885USP2 1767/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.