SCHEMBL14675868

SCHEMBL14675868

O=C(O)C1CN(Cc2ccc(C(F)(F)F)cc2C(F)(F)F)C1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.56
S1PR5 Q9H228 8/20 0.56
GRK5 P34947 1/20 0.56
CDK8 P49336 1/20 0.56
PRKX P51817 1/20 0.54
IKBKE Q14164 1/20 0.54
PDGFRA P16234 2/20 0.53
PIM1 P11309 1/20 0.53
PRKD3 O94806 1/20 0.53
CDK7 P50613 1/20 0.53
JAK3 P52333 1/20 0.53
TNK2 Q07912 1/20 0.53
POLQ O75417 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14779575 0.85 EPHX2 (0.46) S1PR1S1PR5GRK5CDK8PRKX
SCHEMBL14677458 0.81 NR1H2 (0.41) S1PR1S1PR5GRK5CDK8POLQ
SCHEMBL14676489 0.80 NR1H2 (0.40) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL1873186 0.78 S1PR1 (0.58) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL14779622 0.78 NR1H2 (0.39) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL14779624 0.78 NR1H2 (0.39) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL14676460 0.78 NOTUM (0.43) POLQ
SCHEMBL14779566 0.77 NR1H2 (0.39) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL14779564 0.77 NR1H2 (0.39) S1PR1S1PR5PRKXIKBKEPDGFRA
SCHEMBL14675279 0.77 KCNT1 (0.46) PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013018929-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-07 WO disclosed