SCHEMBL14700098

SCHEMBL14700098

CCOc1cccc(COC2CN(c3c4c(nc5ccnn35)CCNCC4)C2)c1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 18/20 0.64
HTR2B P41595 17/20 0.64
HTR2A P28223 16/20 0.64
MAPKAPK2 P49137 1/20 0.34
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10217487 0.92 HTR2C (0.76) HTR2CHTR2BHTR2A
SCHEMBL10218929 0.88 HTR2C (0.82) HTR2CHTR2BHTR2AMAPKAPK2
SCHEMBL2573385 0.86 HTR2C (0.73) HTR2CHTR2BHTR2A
SCHEMBL10217458 0.84 HTR2C (0.70) HTR2CHTR2BHTR2A
SCHEMBL13329044 0.83 HTR2C (0.73) HTR2CHTR2BHTR2AMAPKAPK2
SCHEMBL10219027 0.82 HTR2C (0.80) HTR2CHTR2BHTR2AMAPKAPK2
SCHEMBL10217496 0.81 HTR2C (0.73) HTR2CHTR2BHTR2A
SCHEMBL10218965 0.80 HTR2C (0.81) HTR2CHTR2BHTR2A
SCHEMBL10217493 0.79 HTR2C (0.60) HTR2CHTR2BHTR2A
SCHEMBL10216877 0.79 HTR2C (0.62) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384328-B1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM INT (DE) 2013-02-13 EP disclosed