SCHEMBL14709136

SCHEMBL14709136

CCCSc1nc(Cl)c2nnn(C3CCCC3)c2n1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.58
P2RY12 Q9H244 12/20 0.39
PDE5A O76074 1/20 0.37
PDE1A P54750 1/20 0.37
PDE1B Q01064 1/20 0.37
PDE1C Q14123 1/20 0.37
USP28 Q96RU2 1/20 0.37
ADORA2A P29274 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14709077 0.84 KDM1A (0.44) KDM1AP2RY12
SCHEMBL5729393 0.83 P2RY12 (0.46) KDM1AP2RY12ADORA2A
SCHEMBL5729389 0.83 P2RY12 (0.46) KDM1AP2RY12ADORA2A
SCHEMBL5729958 0.83 P2RY12 (0.46) KDM1AP2RY12ADORA2A
SCHEMBL6075252 0.83 P2RY12 (0.46) KDM1AP2RY12ADORA2A
SCHEMBL21138862 0.83 KDM1A (0.40) KDM1APDE5APDE1APDE1BPDE1C
SCHEMBL5728919 0.79 P2RY12 (0.42) KDM1AP2RY12
SCHEMBL5728911 0.79 P2RY12 (0.42) KDM1AP2RY12
SCHEMBL21268651 0.78 KDM1A (0.44) KDM1APDE5APDE1APDE1BPDE1C
SCHEMBL29385954 0.78 KDM1A (0.44) KDM1APDE5APDE1APDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013023511-A1 TRIAZOLOPYRIMIDINE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF 上海恒瑞医药有限公司 (CN) 2013-02-21 WO disclosed