SCHEMBL14712403

SCHEMBL14712403

Cn1nccc1-c1ccc2c(C(=O)Nc3cnn(Cc4cccc(N)c4)c3)n[nH]c2c1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITK Q08881 16/20 0.62
AURKA O14965 4/20 0.59
RPS6KA3 P51812 1/20 0.47
RPS6KA2 Q15349 1/20 0.47
SCD O00767 2/20 0.43
SCD5 Q86SK9 2/20 0.43
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16163259 0.89 ITK (0.79) ITKAURKASCD
SCHEMBL14712517 0.86 ITK (0.58) ITKAURKARPS6KA3RPS6KA2
SCHEMBL14712567 0.86 ITK (0.60) ITKAURKA
SCHEMBL14712581 0.85 ITK (0.66) ITKAURKA
SCHEMBL14712407 0.85 ITK (0.61) ITKAURKASCDSCD5HCRTR1
SCHEMBL14712518 0.84 ITK (0.63) ITKAURKAHCRTR1HCRTR2
SCHEMBL14712429 0.83 ITK (0.64) ITKAURKA
SCHEMBL14712582 0.82 ITK (0.56) ITKAURKARPS6KA3RPS6KA2
SCHEMBL14712579 0.82 ITK (0.60) ITKAURKA
SCHEMBL14712454 0.81 ITK (0.56) ITKAURKARPS6KA3RPS6KA2SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013024011-A1 INDAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2013-02-21 WO disclosed