SCHEMBL14713170

SCHEMBL14713170

CC#Cc1cncc(C(=O)N=S(C)(=O)c2cccc(C)c2)c1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.57
PDGFRB P09619 11/20 0.57
GRM5 P41594 1/20 0.34
KAT6A Q92794 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL833945 0.91 KDR (0.59) KDRPDGFRBGRM5
SCHEMBL835058 0.91 KDR (0.65) KDRPDGFRBGRM5
SCHEMBL15810261 0.90 KDR (0.61) KDRPDGFRBGRM5
SCHEMBL14713211 0.90 KDR (0.48) KDRPDGFRB
SCHEMBL833621 0.89 KDR (0.57) KDRPDGFRB
SCHEMBL833427 0.89 KDR (0.47) KDRPDGFRBKAT6A
SCHEMBL836724 0.88 KDR (0.59) KDRPDGFRB
SCHEMBL834998 0.88 KDR (0.54) KDRPDGFRB
SCHEMBL836616 0.88 KDR (0.56) KDRPDGFRB
SCHEMBL835190 0.88 KDR (0.56) KDRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099757-B1 SULFOXIMINES AS KINASE INHIBITORS ALLERGAN INC (US) 2014-06-25 EP disclosed
US-8383825-B2 Kinase inhibitors ALLERGAN, INC. (US) 2013-02-26 US disclosed